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DRUG METABOLISM AND PHARMACOKINETICS 27巻 2号

発行元
日本薬物動態学会
ISSN
1347-4367
ISSN(オンライン)
1880-0920
前雑誌
薬物動態

書籍情報から探す
開始頁
The Role of Discovery DMPK Scientists in Industry: Where Do We Go from Here?
Toshiya MORIWAKI
Takeda Pharmaceutical Company Limited
DRUG METABOLISM AND PHARMACOKINETICS 27 (2) 169-170, 2012.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に121円(税込) です。
Quantitative Prediction of Intestinal Glucuronidation of Drugs in Rats Using In Vitro Metabolic Clearance Data
Takako FURUKAWA, Fumihiro NAKAMORI, Kazuhiro TETSUKA, Yoichi NARITOMI, Hiroyuki MORIGUCHI, Katsuhiro YAMANO, Shigeyuki TERASHITA, Toshio TERAMURA
Analysis and Pharmacokinetics Research Laboratories, Astellas Pharma Inc.
DRUG METABOLISM AND PHARMACOKINETICS 27 (2) 171-180, 2012.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
A Practical and Direct Comparison of Intrinsic Metabolic Clearance of Several Non-CYP Enzyme Substrates in Freshly Isolated and Cryopreserved Hepatocytes
Takafumi AKABANE*1,*2, Nicolas GERST*1, Yoichi NARITOMI*2, Jeffrey N.MASTERS*1, Kouichi TAMURA*1
*1Astellas Research Institute of America LLC, *2Analysis and Pharmacokinetics Research Labs, Discovery Drug Metabolism and Pharmacokinetics, Astellas Pharma Inc.
DRUG METABOLISM AND PHARMACOKINETICS 27 (2) 181-191, 2012.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Genetic Polymorphisms in Metabolic and Cellular Transport Pathway of Methotrexate Impact Clinical Outcome of Methotrexate Monotherapy in Japanese Patients with Rheumatoid Arthritis
Tomomi KATO*1, Akinobu HAMADA*1,*2, Shunsuke MORI*3, Hideyuki SAITO*1,*2
*1Department of Clinical Pharmaceutical Sciences, Graduate School of Pharmaceutical Sciences, Kumamoto University, *2Department of Pharmacy, Kumamoto University Hospital, *3Department of Rheumatology, Clinical Research Center for Rheumatic Disease, Kumamoto Saishunso National Hospital
DRUG METABOLISM AND PHARMACOKINETICS 27 (2) 192-199, 2012.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Polycyclic Aromatic Hydrocarbons Activate CYP3A4 Gene Transcription through Human Pregnane X Receptor
Takeshi KUMAGAI*1, Hiroyuki SUZUKI*1, Takamitsu SASAKI*1, Shuhei SAKAGUCHI*1, Shinichi MIYAIRI*2, Yasushi YAMAZOE*3, Kiyoshi NAGATA*1
*1Department of Environmental Health Science, Tohoku Pharmaceutical University, *2Laboratory of Organic Chemistry, School of Pharmacy, Nihon University, *3Division of Drug Metabolism and Molecular Toxicology, Graduate School of Pharmaceutical Sciences, Tohoku University
DRUG METABOLISM AND PHARMACOKINETICS 27 (2) 200-206, 2012.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
The Pharmacokinetic-pharmacodynamic Assessment of the Hypotensive Effect after Coadministration of Losartan and Hydrochlorothiazide in Spontaneously Hypertensive Rats
Ryosuke SHIMIZU*1,*2, Makoto MIYAZAKI*2, Kazunori IWANAGA*2, Masawo KAKEMI*2
*1Drug Metabolism & Pharmacokinetics, Drug Developmental Research Laboratories, Shionogi & Co.,Ltd., *2Division of Pharmaceutics, Osaka University of Pharmaceutical Sciences
DRUG METABOLISM AND PHARMACOKINETICS 27 (2) 207-215, 2012.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Pharmacokinetics and Pharmacodynamics of KR-66223, a Novel DPP-4 Inhibitor
Jin Sook SONG*1, Kyeong-Ryoon LEE*1, Hyun Jin KWON*1, Sang Dal RHEE*2, Min Sun KIM*1, Sung Hum CHOI*1, Sung-Hack LEE*4, Im Sook SONG*3, Jin Hee AHN*2, Sung Hoon AHN*1, Myung Ae BAE*1
*1Drug Discovery Platform Technology Team, Division of Bio-organic Science, Korea Research Institute of Chemical Technology, *2Bio-Organic Science Division, Korea Research Institute of Chemical Technology, *3Department of Pharmacology and Pharmacogenomics Research Center, Inje University College of Medicine, *4Drug Metabolism and Pharmacokinetics Department, LG Life Sciences R&D
DRUG METABOLISM AND PHARMACOKINETICS 27 (2) 216-222, 2012.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Metabolic Fate of Sipoglitazar, a Novel Oral PPAR Agonist with Activities for PPAR-γ,-α and -δ, in Rats and Monkeys and Comparison with Humans In Vitro
Mitsuhiro NISHIHARA, Miyako SUDO, Hidenori KAMIGUCHI, Naohiro KAWAGUCHI, Yoshihiro MAESHIBA, Yutaka KIYOTA, Junzo TAKAHASHI, Yoshihiko TAGAWA, Takahiro KONDO, Satoru ASAHI
Drug Metabolism and Pharmacokinetics Research Laboratories, Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited
DRUG METABOLISM AND PHARMACOKINETICS 27 (2) 223-231, 2012.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Peptide Cotransporter 1 in Intestine and Organic Anion Transporters in Kidney Are Targets of Interaction between JBP485 and Lisinopril in Rats
Xinjin GUO*1, Qiang MENG*1,*3, Qi LIU*1,*3, Changyuan WANG*1,*3, Qi MAO*1, Huijun SUN*1,*3, Jinyong PENG*1,*3, Taiichi KAKU*2, Kexin LIU*1,*3
*1Department of Clinical Pharmacology, College of Pharmacy, Dalian Medical University, *2Japan Bioproducts Industry Co.Ltd., *3Provincial Key Laboratory for Pharmacokinetics and Transport, Liaoning, Dalian Medical University
DRUG METABOLISM AND PHARMACOKINETICS 27 (2) 232-241, 2012.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Food-drug Interaction of Tacrolimus with Pomelo, Ginger, and Turmeric Juice in Rats
Kanoko EGASHIRA*1,*2, Hitoshi SASAKI*1, Shun HIGUCHI*3, Ichiro IEIRI*2
*1Department of Hospital Pharmacy, Nagasaki University Hospital, *2Department of Clinical Pharmacokinetics, Graduate School of Pharmaceutical Science, Kyushu University, *3Academic, Industrial and Governmental Liaison Center, Fukuoka University
DRUG METABOLISM AND PHARMACOKINETICS 27 (2) 242-247, 2012.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Impact of Concomitant Antacid Administration on Gabapentin Plasma Exposure and Oral Bioavailability in Healthy Adult Subjects
Tatsuya YAGI*1, Takafumi NAITO*1, Yasuaki MINO*1, Kazuo UMEMURA*2, Junichi KAWAKAMI*1
*1Department of Hospital Pharmacy, Hamamatsu University School of Medicine, *2Department of Pharmacology, Hamamatsu University School of Medicine
DRUG METABOLISM AND PHARMACOKINETICS 27 (2) 248-254, 2012.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Nicotinate Uptake by Two Kinetically Distinct Na+ -Dependent Carrier-Mediated Transport Systems in the Rat Small Intestine
Masahiko OHKUBO, Kinya OHTA, Katsuhisa INOUE, Hiroaki YUASA
Department of Biopharmaceutics, Graduate School of Pharmaceutical Sciences, Nagoya City University
DRUG METABOLISM AND PHARMACOKINETICS 27 (2) 255-262, 2012.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
An Artifact Derived from a Pseudogene Led to the Discovery of MicroRNA Binding Site Polymorphism in the 3'-Untranslated Region of the Human Dihydrofolate Reductase Gene
Hideki HAYASHI*1, Yui TAZOE*1, Masato HORINO*1, Chihiro FUJIMAKI-KATOH*1, Seiji TSUBOI*2, Taiji MATSUYAMA*3, Kazuhiro KOSUGE*4, Hiroshi YAMADA*4, Daiki TSUJI*1, Kazuyuki INOUE*1, Kunihiko ITOH*1
*1Department of Clinical Pharmacology & Genetics, School of Pharmaceutical Sciences, University of Shizuoka, *2Department of Rheumatology, Shizuoka Kousei Hospital, *3Department of Pharmacy, Shizuoka Kousei Hospital, *4Department of Drug Evaluation & Informatics, School of Pharmaceutical Sciences, University of Shizuoka
DRUG METABOLISM AND PHARMACOKINETICS 27 (2) 263-267, 2012.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
An Evaluation of Single Nucleotide Polymorphisms in the Human Heat Shock Protein 90 kDa Alpha and Beta Isoforms
Jonathan D.URBAN*1, Robert A.BUDINSKY*2, J.Craig ROWLANDS*2
*1ToxStrategies, *2The Dow Chemical Company, Toxicology and Environmental Research and Consulting
DRUG METABOLISM AND PHARMACOKINETICS 27 (2) 268-278, 2012.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。