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Chemical & Pharmaceutical Bulletin 58巻 8号

発行元
日本薬学会
ISSN
0009-2363
ISSN(オンライン)
1347-5223

書籍情報から探す
開始頁
Synthesis, Characterization, Cytotoxic Activities, and DNA-Binding Studies of Ternary Copper(II) Complexes with New Coumarin Derivatives
Lei JIAa,b, Xi-Ming XUc, Jun XUa, Long-Hai CHENa, Peng JIANGc, Fei-Xiang CHENGa, Guang-Nong LUa, Qin WANGc, Jin-Cai WUa, Ning TANGa
aKey Laboratory of Nonferrous Metal Chemistry and Resources Utilization of Gansu Province, State Key Laboratory of Applied Organic Chemistry, College of Chemistry and Chemical Engineering, Lanzhou University, bDepartment of Physics and Chemistry, Henan Polytechnic University, cSchool of Life Science, Lanzhou University
Chemical & Pharmaceutical Bulletin 58 (8) 1003-1008, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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A New Method for Evaluating the Bitterness of Medicines in Development Using a Taste Sensor and a Disintegration Testing Apparatus
Tsutomu HARADAa, Takahiro UCHIDAb, Miyako YOSHIDAb, Yoshikazu KOBAYASHIc, Ryuichi NARAZAKId, Takayuki OHWAKIe
aPlanning & Operations Section, Customer Joy Department, CEO office, Eisai Co.,Ltd., bSchool of Pharmaceutical Sciences, Mukogawa Women's University, cIntelligent Sensor Technology, Inc., dFormulation Research, CMC Japan, Pharmaceutical Science and Technology CFU, Eisai Co.,Ltd., eDrug Development Technology Center, Customer Joy Department, CEO Office, Eisai Co.,Ltd.
Chemical & Pharmaceutical Bulletin 58 (8) 1009-1014, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Preparation and the in Vitro Evaluation of Nanoemulsion System for the Transdermal Delivery of Granisetron Hydrochloride
Wen-wu ZHENGa, Ling ZHAOb, Yu-meng WEIb, Yun YEb, Shun-han XIAOb
aDepartment of Cardiology, the People's Hospital of Luzhou, bDepartment of Pharmaceutics, School of Pharmacy, Luzhou Medical College
Chemical & Pharmaceutical Bulletin 58 (8) 1015-1019, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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1-(3'-[125I]Iodophenyl)-3-methy-2-pyrazolin-5-one: Preparation, Solution Stability, and Biodistribution in Normal Mice
Yuuhei SANO, Tomokazu MOTOMURA, Fumihiko YAMAMOTO, Miki FUKUDA, Takahiro MUKAI, Minoru MAEDA
Graduate School of Pharmaceutical Sciences, Kyushu University
Chemical & Pharmaceutical Bulletin 58 (8) 1020-1025, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Crotalionosides A―C, Three New Megastigmane Glucosides, Two New Pterocarpan Glucosides and a Chalcone C-Glucoside from the Whole Plants of Crotalaria zanzibarica
Junko SHITAMOTOa, Katsuyoshi MATSUNAMIa, Hideaki OTSUKAa, Takakazu SHINZATOb, Yoshio TAKEDAc
aDepartment of Pharmacognosy, Graduate School of Biomedical Sciences, Hiroshima University, bSubtropical Field Science Center, Faculty of Agriculture, University of the Ryukyus, cFaculty of Pharmacy, Yasuda Women's University
Chemical & Pharmaceutical Bulletin 58 (8) 1026-1032, 2010.
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Azaphilone and Isocoumarin Derivatives from the Endophytic Fungus Penicillium sclerotiorum PSU-A13
Jiraporn ARUNPANICHLERTa, Vatcharin RUKACHAISIRIKULa, Yaowapa SUKPONDMAa, Souwalak PHONGPAICHITb, Supinya TEWTRAKULc, Nuttawut RUNGJINDAMAId, Jariya SAKAYAROJd
aDepartment of Chemistry and Center for Innovation in Chemistry, Faculty of Science, Prince of Songkla University, bNatural Products Research Center and Department of Microbiology, Faculty of Science, Prince of Songkla University, cDepartment of Pharmacognosy and Pharmaceutical Botany, Faculty of Pharmaceutical Sciences, Prince of Songkla University, dNational Center for Genetic Engineering and Biotechnology (BIOTEC)
Chemical & Pharmaceutical Bulletin 58 (8) 1033-1036, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Development and in Vitro Evaluation of Ibuprofen Mouth Dissolving Tablets Using Solid Dispersion Technique
Sunil Kumar JAINa, Meenakshi SHUKLAb, Vivek SHRIVASTAVAc
aSLT Institute of Pharmaceutical Sciences, Guru Ghasidas Vishwavidyalaya, bBansal College of Pharmacy, cBhopal Institute of Technology and Science-Pharmacy
Chemical & Pharmaceutical Bulletin 58 (8) 1037-1042, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Dolabellane Diterpene and Three Cycloartane Glycosides from Thalictrum squarrosum
Hitoshi YOSHIMITSUa, Hiroyuki MIYASHITAa, Makiko NISHIDAb, Tomoko MINENOc, Toshihiro NOHARAa
aFaculty of Pharmaceutical Sciences, Sojo University, bFaculty of Home Economics, Kyushu Women's University, cFaculty Pharmacy, Takasaki University of Health and Welfare
Chemical & Pharmaceutical Bulletin 58 (8) 1043-1046, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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In Vitro Leishmanicidal Activity of Benzophenanthridine Alkaloids from Bocconia pearcei and Related Compounds
Hiroyuki FUCHINOa, Marii KAWANOb, Kanami MORI-YASUMOTOc, Setsuko SEKITAc, Motoyoshi SATAKEd, Tsutomu ISHIKAWAe, Fumiyuki KIUCHIf, Nobuo KAWAHARAa
aResearch Center for Medicinal Plant Resources, National Institute of Biomedical Innovation, bFaculty of Pharmaceutical Sciences, Josai International University, cDepartment of Pharmaceutical Technology, Faculty of Pharmaceutical Sciences at Kagawa Campus, Tokushima Bunri University, dInstitute of Environmental Science for Human Life, Ochanomizu University, eFaculty of Pharmaceutical Sciences, Chiba University, fFaculty of Pharmacy, Keio University
Chemical & Pharmaceutical Bulletin 58 (8) 1047-1050, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Evaluation of Serum Protein Binding by Using in Vitro Pharmacological Activity for the Effective Pharmacokinetics Profiling in Drug Discovery
Yukinori KAWAI, Yoshimine FUJII, Katsuya AKIMOTO, Masayuki TAKAHASHI
Drug Metabolism & Pharmacokinetics Research Laboratories, Daiichi Sankyo Co.,Ltd.
Chemical & Pharmaceutical Bulletin 58 (8) 1051-1056, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Novel Acyl-CoA: Cholesterol Acyltransferase Inhibitor: Indoline-Based Sulfamide Derivatives with Low Lipophilicity and Protein Binding Ratio
Kenji TAKAHASHI, Masaru OHTA, Yoshimichi SHOJI, Masayasu KASAI, Kazuyoshi KUNISHIRO, Tomohiro MIIKE, Mamoru KANDA, Hiroaki SHIRAHASE
Research Laboratories, Kyoto Pharmaceutical Industries, Ltd.
Chemical & Pharmaceutical Bulletin 58 (8) 1057-1065, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Novel Tetrahydroisoquinoline Derivatives with Inhibitory Activities against Acyl-CoA: Cholesterol Acyltransferase and Lipid Peroxidation
Masaru OHTAa,b, Kenji TAKAHASHIa, Masayasu KASAIa, Yoshimichi SHOJIa, Kazuyoshi KUNISHIROa, Tomohiro MIIKEa, Mamoru KANDAa, Chisato MUKAIb, Hiroaki SHIRAHASEa
aReseareh Laboratories, Kyoto Pharmaceutical Industries, Ltd., bDivision of Pharmaceutical Sciences, Graduate School of Natural Science and Technology, Kanazawa University
Chemical & Pharmaceutical Bulletin 58 (8) 1066-1076, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Synthesis, Crystal Structure, Antioxidant Activity, and DNA-Binding Studies of a Novel Ni(II) [2×2] Grid Complex with a Rigid Bistridentate Schiff Base Ligand
Lei JIAa,b, Jun XUa, Xi-Ming XUc, Long-Hai CHENa, Peng JIANGc, Fei-Xiang CHENGa, Guang-Nong LUa, Qin WANGc, Jin-Cai WUa, Ning TANGa
aKey Laboratory of Nonferrous Metal Chemistry and Resources Utilization of Gansu Province, State Key Laboratory of Applied Organic Chemistry, College of Chemistry and Chemical Engineering, Lanzhou University, bDepartment of Physics and Chemistry, Henan Polytechnic University, cSchool of Life Science, Lanzhou University
Chemical & Pharmaceutical Bulletin 58 (8) 1077-1080, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Synthesis and Antibacterial Activity of Some Novel 6-(1H-Benz[d]imidazol-2-yl)-8-(5-nitro-2-furyl)-3-(4-pyridyl)-7,8-dihydro[1,2,4]triazolo[3,4-b][1,3,4]thiadiazepines
Vanga MALLA REDDY, Kunduru RAVINDER REDDY
Ch.Ravishanker Memorial Medicinal Chemistry Research Laboratory, University College of Pharmaceutical Sciences, Kakatiya University
Chemical & Pharmaceutical Bulletin 58 (8) 1081-1084, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Oppositinines A and B: New Vasorelaxant β-Carboline Alkaloids from Neisosperma oppositifolia
Kartini AHMADa, Noel F.THOMASb, A.Hamid A.HADIb, Mat Ropi MUKHTARb, Khalit MOHAMADc, Mohd Azlan NAFIAHa, Koichi TAKEYAd, Hiroshi MORITAe, Marc LITAUDONf, Hiroko ARAIe, Khalijah AWANGb
aDepartment of Chemistry, Faculty of Science and Technology, University Pendidikan Sultan Idris, bDepartment of Chemistry, Faculty of Science, University of Malaya, cDepartment of Pharmacy, Faculty of Medicine, University of Malaya, dTokyo University of Pharmacy and Life Sciences, eFaculty of Pharmaceutical Sciences, Hoshi University, fInstitut de Chimie des Substances Naturelles
Chemical & Pharmaceutical Bulletin 58 (8) 1085-1087, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Three New Cardenolides from Methanol Extract of Stems and Twigs of Nerium oleander
Liming BAIa, Ming ZHAOa, Asami TOKIb, Jun-ichi SAKAIc, Xiao-yang YANGd, Yuhua BAIe, Mariko ANDOf, Katsutoshi HIROSEg, Masayoshi ANDOc
aCollege of Chemistry and Chemistry Engineering, Qiqihar University, bGraduate School of Science and Technology, Niigata University, cDepartment of Chemistry and Chemical Engineering, Faculty of Engineering, Niigata University, dAtmospheric Chemistry & Aerosol Division, Chinese Research Academy of Environmental Science, eDepartment of Medicinal Chemistry, Pharmaceutical Department, Daqing Campus of Harbin Medical University, fTechnical Division, School of Engineering, Tohoku University, gKNC Laboratories Co.,Ltd.
Chemical & Pharmaceutical Bulletin 58 (8) 1088-1092, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Two New Aristolochic Acid Derivatives from the Roots of Aristolochia fangchi and Their Cytotoxicities
Yu CAIa, Tian-Ge CAIb
aSchool of Pharmacy, Jinan University, bSchool of Life Science, Liaoning University
Chemical & Pharmaceutical Bulletin 58 (8) 1093-1095, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Effect of Particle Size on Skin Permeation and Retention of Piroxicam in Aqueous Suspension
Kunikazu MORIBEa, Mizuho SHIBATAa, Takayuki FURUISHIb, Kenjirou HIGASHIa, Kazuo TOMONOb, Keiji YAMAMOTOa
aGraduate School of Pharmaceutical Sciences, Chiba University, bResearch Unit of Pharmaceutics, School of Pharmacy, Nihon University
Chemical & Pharmaceutical Bulletin 58 (8) 1096-1099, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Triterpenoid Derivatives from Cylicodiscus gabunensis
Pierre MKOUNGAa, Alembert Tchinda TIABOUb, Jacques KOUAMa
aDepartment of Organic Chemistry, Faculty of Sciences, University of Yaounde I, bInstitute of Medical Research and Medicinal Plants Studies (IMPM)
Chemical & Pharmaceutical Bulletin 58 (8) 1100-1102, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Chemical Synthesis of (22E)-3α,6α,7α,12α-Tetrahydroxy-5β-chol-22-en-24-oic Acid and Its N-Acylamidated Conjugates with Glycine or Taurine: Precursors of the [22,23-3H] Labelled Tracers
Shoujiro OGAWAa, Yuuki ADACHIa, Genta KAKIYAMAa, Miki SHIMADAb, Nariyasu MANOb, Junichi GOTOb, Takashi IIDAa
aDepartment of Chemistry, College of Humanities & Sciences, Nihon University, bDepartment of Pharmaceutical Sciences, Tohoku University Hospital
Chemical & Pharmaceutical Bulletin 58 (8) 1103-1106, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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An Effective Synthesis of 5,4'-Disubstituted Flavones via a Cesium Enolate Assisted Intramolecular ipso-Substitution Reaction
Masato MATSUGI, Masaki TAKEDA, Ayano TAKAHASHI, Takahide TAZAKI, Hiroto TAMURA, Takayuki SHIOIRI
Department of Applied Biological Chemistry, Faculty of Agriculture, Meijo University
Chemical & Pharmaceutical Bulletin 58 (8) 1107-1110, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Steamed Ginseng-Leaf Components Enhance Cytotoxic Effects on Human Leukemia HL-60 Cells
Nguyen Huu TUNGa,b, Gyu Yong SONGa, Chau Van MINHb, Phan Van KIEMb, Long Guo JINa, Hye-Jin BOOc, Hee-Kyoung KANGc, Young Ho KIMa
aCollege of Pharmacy, Chungnam National University, bInstitute of Natural Products Chemistry, Vietnam Academy of Science and Technology, cDepartment of Pharmacology, School of Medicine, Institute of Medical Sciences, Jeju National University
Chemical & Pharmaceutical Bulletin 58 (8) 1111-1115, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Cucullamide, a New Putrescine Bisamide from Amoora cucullata
Mohamed Saleh ABDELFATTAHa,c, Kazufumi TOUMEa, Firoj AHMEDa,b, Samir Kumar SADHUb, Masami ISHIBASHIa
aGraduate School of Pharmaceutical Sciences, Chiba University, bPharmacy Discipline, Life Science School, Khulna University, cChemistry Department, Faculty of Science, Helwan University
Chemical & Pharmaceutical Bulletin 58 (8) 1116-1118, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Structures of New Erythrinan Alkaloids and Nitric Oxide Production Inhibitors from Erythrina crista-galli
Masaaki OZAWAa, Shunsuke KAWAMATAb, Tadahiro ETOHc, Masahiko HAYASHIc, Kanki KOMIYAMAd, Akio KISHIDAa, Chiaki KURODAb, Ayumi OHSAKIa
aInstitute of Biomaterials and Bioengineering, Tokyo Medical and Dental University, bDeparment of Chemistry, Rikkyo University, cFaculty of Pharmacy, Iwaki Meisei University, dKitasato Research Center of Environmental Science, Kitasato University
Chemical & Pharmaceutical Bulletin 58 (8) 1119-1122, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Antibacterial Activity of 5-Dialkylaminomethylhydantoins and Related Compounds
Fumiko FUJISAKI, Kaori SHOJI, Mari SHIMODOUZONO, Nobuhiro KASHIGE, Fumio MIAKE, Kunihiro SUMOTO
Faculty of Pharmaceutical Science, Fukuoka University
Chemical & Pharmaceutical Bulletin 58 (8) 1123-1126, 2010.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。