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Chemical & Pharmaceutical Bulletin 59巻 8号

発行元
日本薬学会
ISSN
0009-2363
ISSN(オンライン)
1347-5223

書籍情報から探す
開始頁
Synthesis and Evaluation of Analgesic and Anti-inflammatory Activities of Most Active Free Radical Scavenging Derivatives of Embelin -A Structure-Activity Relationship
Sekar MAHENDRANa, Shrishailappa BADAMIb, Subban RAVIc, Boreddy Shivanandappa THIPPESWAMYb, Veeresh Prabhakar VEERAPURb
aDepartment of Pharmaceutical Chemistry, J.S.S.College of Pharmacy, bSree Siddaganga College of Pharmacy, cDepartment of Chemistry, Karpagam University
Chemical & Pharmaceutical Bulletin 59 (8) 913-919, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Formulation and Optimization of Orally Disintegrating Tablets of Sumatriptan Succinate
Ravi SHESHALAa,b, Nurzalina KHANa, Yusrida DARWISa
aSchool of Pharmaceutical Sciences, Universiti Sains Malaysia, bSchool of Pharmacy and Health Sciences, International Medical University
Chemical & Pharmaceutical Bulletin 59 (8) 920-928, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Optimization and Characterization of Dry Powder of Fanhuncaoin for Inhalation Based on Selection of Excipients
Xiao-bo YANGa, Xiao-bo WANGa,b, Wei-san PANa, Rong-gang XIb, Yi-nan WANGc, Dan LIUb, Yan SHIb, Shuang JIANGb
aDepartment of Pharmaceutics, Shenyang Pharmaceutical University, bThe 210th Hospital of PLA, cThe First Affiliated Hospital of Dalian Medical University
Chemical & Pharmaceutical Bulletin 59 (8) 929-937, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
11C-Labeled Analogs of Indomethacin Esters and Amides for Brain Cyclooxygenase-2 Imaging: Radiosynthesis, in Vitro Evaluation and in Vivo Characteristics in Mice
Yumi YAMAMOTOa, Jun TOYOHARAb, Kiichi ISHIWATAb, Kohei SANOa, Fumihiko YAMAMOTOa, Takahiro MUKAIa,c, Minoru MAEDAa
aGraduate School of Pharmaceutical Sciences, Kyushu University, bPositron Medical Center, Tokyo Metropolitan Institute of Gerontology, cKobe Pharmaceutical University
Chemical & Pharmaceutical Bulletin 59 (8) 938-946, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Bisbenzylisoquinoline Alkaloids from Nelumbo nucifera
Atsuko ITOHa, Tomomi SAITOHa, Kaori TANIa, Misaki UCHIGAKIa, Yumi SUGIMOTOb, Jun YAMADAb, Hiroshi NAKAJIMAc, Hideo OHSHIROd, Schujian SUNd, Takao TANAHASHIa
aKobe Pharmaceutical University, bYokohama College of Pharmacy, cResearch Center for Industry Innovation, Osaka City University, dShanghai University of Traditional Chinese Medicine
Chemical & Pharmaceutical Bulletin 59 (8) 947-951, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
In Vitro Evaluation of Mucoadhesive Vaginal Tablets of Antifungal Drugs Prepared with Thiolated Polymer and Development of a New Dissolution Technique for Vaginal Formulations
Esra BALOGLUa, Zeynep AY SENYIGITa, Sinem Yaprak KARAVANAa, Anja VETTERb, Dilek Yesim METINc, Suleyha HILMIOGLU POLATc, Tamer GUNERIa, Andreas BERNKOP-SCHNURCHb
aDepartment of Pharmaceutical Technology, Faculty of Pharmacy, Ege University, bDepartment of Pharmaceutical Technology, Institute of Pharmacy, University of Innsbruck, cDepartment of Microbiology and Clinical Microbiology, Faculty of Medicine, Ege University
Chemical & Pharmaceutical Bulletin 59 (8) 952-958, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Formulation Study for Orally Disintegrating Tablet Using Partly Pregelatinized Starch Binder
Kazuki MIMURAa,b, Ken KANADAb, Shinya UCHIDAa, Masaki YAMADAb, Noriyuki NAMIKIa
aDepartment of Pharmacy Practice and Science, School of Pharmaceutical Sciences University of Shizuoka, bPharmaceutical Research & Development, Kissei Pharmaceutical Co., Ltd.
Chemical & Pharmaceutical Bulletin 59 (8) 959-964, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Metal-Binding Ability of Human Prion Protein Fragment Peptides Analyzed by Column Switch HPLC
Aya KOJIMA, Yasunori MABUCHI, Motomi KONISHI, Rika OKIHARA, Makoto NAGANO, Toshifumi AKIZAWA
Department of Analytical Chemistry, Pharmaceutical Science, Setsunan University
Chemical & Pharmaceutical Bulletin 59 (8) 965-971, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Oral Administration of Bis(aspirinato)zinc(II) Complex Ameliorates Hyperglycemia and Metabolic Syndrome-Like Disorders in Spontaneously Diabetic KK-Ay Mice: Structure-Activity Relationship on Zinc-Salicylate Complexes
Yutaka YOSHIKAWAa, Yusuke ADACHIa, Hiroyuki YASUIa, Masakazu HATTORIb, Hiromu SAKURAIc
aDepartment of Analytical and Bioinorganic Chemistry, Kyoto Pharmaceutical University, bDivision of Diabetes, Clinical Research Institute for Endocrine and Metabolic Diseases, National Hospital Organization, Kyoto Medical Center, cDepartment of Pharmaco-analytical and Biocoordination Chemistry, Faculty of Pharmaceutical Sciences, Suzuka University of Medical Science
Chemical & Pharmaceutical Bulletin 59 (8) 972-977, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Synthesis and Characterization of Two Homologous Series of Diastereomeric 2-Alkoxyphenylcarbamates
Fridrich GREGANa, Juraj GREGANb, Marek SKORSEPAa
aDepartment of Chemistry, Faculty of Natural Sciences, Matej Bel University, bMax F.Perutz Laboratories, Department of Chromosome Biology, University of Vienna
Chemical & Pharmaceutical Bulletin 59 (8) 978-983, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Design, Synthesis and Antitumor Activity of Novel Artemisinin Derivatives Using Hybrid Approach
Lijun XIEa, Xin ZHAIa, Lixiang RENb, Haiyan MENGa, Chun LIUa, Wufu ZHUa, Yanfang ZHAOa
aKey Laboratory of Original New Drug Design and Discovery of Ministry of Education, Shenyang Pharmaceutical University, bShenyang J & Health Bio-technic Development Co., Ltd.
Chemical & Pharmaceutical Bulletin 59 (8) 984-990, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Discovery of Novel Thieno[2,3-d]pyrimidin-4-yl Hydrazone-Based Cyclin-Dependent Kinase 4 Inhibitors: Synthesis, Biological Evaluation and Structure-Activity Relationships
Takao HORIUCHIa, Yasuyuki TAKEDAa, Noriyasu HAGINOYAa, Masaki MIYAZAKIa, Motoko NAGATAb, Mayumi KITAGAWAb, Kouichi AKAHANEb, Kouichi UOTOa
aLead Discovery & Optimization Research Laboratories II, Daiichi Sankyo Co., Ltd., bOncology Research Laboratories, Daiichi Sankyo Co., Ltd.
Chemical & Pharmaceutical Bulletin 59 (8) 991-1002, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Limonoids and Triterpenoids from the Seeds of Melia azedarach
Hong-Bing LIU, Chuan-Rui ZHANG, Shi-Hui DONG, Lei DONG, Yan WU, Jian-Min YUE
State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences
Chemical & Pharmaceutical Bulletin 59 (8) 1003-1007, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Configurational Studies of Complexes of Various Tea Catechins and Caffeine in Crystal State
Hiroyuki TSUTSUMI, Yoshifumi KINOSHITA, Takashi SATO, Takashi ISHIZU
Faculty of Pharmacy and Pharmaceutical Sciences, Fukuyama University
Chemical & Pharmaceutical Bulletin 59 (8) 1008-1015, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Synthesis and Antiviral Activity of Novel 1,3,4-Thiadiazine Derivatives
Yajun YANGa,b, Ziming FENGa, Jianshuang JIANGa, Yanan YANGa, Xiandao PANa,c, Peicheng ZHANGa
aKey Laboratory of Bioactive Substances and Resources Utilization of Chinese Herbal Medicine (Ministry of Education), Institute of Materia Medica, Chinese Academy of Medical Sciences and Peking Union Medical College, bKey Laboratory of Human Disease Comparative Medicine, Ministry of Health, Institute of Laboratory Animal Science, Chinese Academy of Medical Sciences & Comparative Medical Center, Peking Union Medical College, cBeijing Union Pharmaceutical Factory
Chemical & Pharmaceutical Bulletin 59 (8) 1016-1019, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Chemical Structures and Hepatoprotective Effects of Constituents from the Leaves of Salacia chinensis
Seikou NAKAMURAa, Yi ZHANGa, Hisashi MATSUDAa, Kiyofumi NINOMIYAb, Osamu MURAOKAb, Masayuki YOSHIKAWAa
aKyoto Pharmaceutical University, bPharmaceutical Research and Technology Institute, Kinki University
Chemical & Pharmaceutical Bulletin 59 (8) 1020-1028, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Synthesis and Pharmacological Evaluation of 1-Isopropyl-1,2,3,4-tetrahydroisoquinoline Derivatives as Novel Antihypertensive Agents
Susumu WATANUKIa, Keisuke MATSUURAa, Yuichi TOMURAa, Minoru OKADAb, Toshio OKAZAKIc, Mitsuaki OHTAa, Shin-ichi TSUKAMOTOa
aDrug Discovery Research, Astellas Pharma Inc., bTechnology, Astellas Pharma Inc., cQA, RA and Pharmacovigilance, Astellas Pharma Inc.
Chemical & Pharmaceutical Bulletin 59 (8) 1029-1037, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Biotransformation of a Taxadiene by Ginkgo Cell Cultures and the Tumor Multi-Drug Resistant Reversal Activities of the Metabolites
Dan XIE, Yi ZHANG, Jianhua ZOU, Dali YIN, Xiaoguang CHEN, Jungui DAI
State Key Laboratory of Bioactive Substances and Functions of Natural Medicines, Institute of Materia Medica, Chinese Academy of Medical Sciences & Peking Union Medical College
Chemical & Pharmaceutical Bulletin 59 (8) 1038-1041, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Microbial Conversion of Curcumin into Colorless Hydroderivatives by the Endophytic Fungus Diaporthe sp. Associated with Curcuma longa
Shoji MAEHARAa, Michiteru IKEDAa, Hiroyuki HARAGUCHIb, Chinami KITAMURAa, Tetsuro NAGOEc, Kazuyoshi OHASHIa, Hirotaka SHIBUYAa
aFaculty of Pharmacy and Pharmaceutical Sciences, Fukuyama University, bFaculty of Life Science and Biotechnology, Fukuyama University, cRohokeimeido Co., Ltd.
Chemical & Pharmaceutical Bulletin 59 (8) 1042-1044, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Synthesis and Biological Evaluation of Two Salidroside Analogues in the PC12 Cell Model Exposed to Hypoglycemia and Serum Limitation
Yibing GUOa,b,c, Xiaohong LIa, Yahong ZHAOb, Yongxing SIb, Hui ZHUa, Yumin YANGb
aSurgical Comprehensive Laboratory of Affiliated Hospital, Nantong University, bJiangsu Key Laboratory of Neuroregeneration, Nantong University, cMedical School, Nantong University
Chemical & Pharmaceutical Bulletin 59 (8) 1045-1047, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
(-)-Hydroxylindestrenolide, a New Sesquiterpenoid from a Gorgonian Coral Menella sp. (Plexauridae)
Shih-Yao KAOa,b, Yu-Chia CHANGb,c, Jui-Hsin SUa,b, Mei-Chin LUa,b, Yung-Husan CHENb, Jyh-Horng SHEUd,e, Zhi-Hong WENd,e, Wei-Hsien WANGb,d,e, Yueh-Hsiung KUOf, Tsong-Long HWANGg, Ping-Jyun SUNGa,b,d,e,h
aGraduate Institute of Marine Biotechnology, National Dong Hwa University, bNational Museum of Marine Biology and Aquarium, cDoctoral Degree Program in Marine Biotechnology, National Sun Yat-sen University and Academia Sinica, dDepartment of Marine Biotechnology and Resources, National Sun Yat-sen University, eDivision of Marine Biotechnology, Asia-Pacific Ocean Research Center, National Sun Yat-sen University, fTsuzuki Institute for Traditional Medicine, College of Pharmacy, China Medical University, gGraduate Institute of Natural Products, Chang Gung University, hDepartment of Life Science and Institute of Biotechnology, National Dong Hwa University
Chemical & Pharmaceutical Bulletin 59 (8) 1048-1050, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Synthesis of New α-Glucosidase Inhibitors Based on Oleanolic Acid Incorporating Cinnamic Amides
Wei NIEa, Jian-Guang LUOa, Xiao-Bing WANGa, Hong YINa, Hong-Bin SUNb, He-Quan YAOb, Ling-Yi KONGa
aDepartment of Natural Medicinal Chemistry, China Pharmaceutical University, bDepartment of Medicinal Chemistry, China Pharmaceutical University
Chemical & Pharmaceutical Bulletin 59 (8) 1051-1056, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Synthesis, Cytotoxicities and DNA-Binding Affinities of Benzofuran-3-ols and Their Fused Analogs
Zhong-Zhen ZHOUa, Min ZOUa, Jia ZHOUa, Chun-Qiong ZHOUa, Yan-Hong DENGa, Ming-Hui CHENa, Chun-Ping GUa, Zhi-Hong JIANGa,b, Wen-Hua CHENa, Shu-Wen LIUa
aSchool of Pharmaceutical Sciences, Southern Medical University, bSchool of Chinese Medicine, Hong Kong Baptist University
Chemical & Pharmaceutical Bulletin 59 (8) 1057-1061, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Efficient Synthesis of [11C]Ramelteon as a Positron Emission Tomography Probe for Imaging Melatonin Receptors Involved in Circadian Rhythms
Misato TAKASHIMA-HIRANO, Syusaku TAZAWA, Kazuhiro TAKAHASHI, Hisashi DOI, Masaaki SUZUKI
RIKEN Center for Molecular Imaging Science (CMIS)
Chemical & Pharmaceutical Bulletin 59 (8) 1062-1064, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Four New Iridoid Glucosides from Ajuga reptans
Masateru ONOa, Chisato FURUSAWAa, Takumi OZONOa, Keisuke ODAa, Shin YASUDAa, Masafumi OKAWAb, Junei KINJOb, Tsuyoshi IKEDAc, Hiroyuki MIYASHITAc, Hitoshi YOSHIMITSUc, Toshihiro NOHARAc
aTokai University School of Agriculture, bFaculty of Pharmaceutical Sciences, Fukuoka University, cFaculty of Pharmaceutical Sciences, Sojo University
Chemical & Pharmaceutical Bulletin 59 (8) 1065-1068, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Synthesis of N-[2-(2,4-Difluorophenoxy)trifluoromethyl-3-pyridyl]sulfonamides and Their Inhibitory Activities against Secretory Phospholipase A2
Hitoshi NAKAYAMAc, Keiichi ISHIHARAb, Satoshi AKIBAb, Jun'ichi UENISHIa
aDepartment of Pharmaceutical Chemistry, Kyoto Pharmaceutical University, bDepartment of Pathological Biochemistry, Kyoto Pharmaceutical University, cOrganic Chemicals Division, R/D Strategy Headquarters, Ishihara Sangyo Kaisha
Chemical & Pharmaceutical Bulletin 59 (8) 1069-1072, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Cinchona Alkaloids Are Also Produced by an Endophytic Filamentous Fungus Living in Cinchona Plant
Shoji MAEHARAa, Partomuan SIMANJUNTAKb, Chinami KITAMURAa, Kazuyoshi OHASHIa, Hirotaka SHIBUYAa
aFaculty of Pharmacy and Pharmaceutical Sciences, Fukuyama University, bResearch Center for Biotechnology, Indonesian Institute of Sciences
Chemical & Pharmaceutical Bulletin 59 (8) 1073-1074, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に121円(税込) です。
Synthesis and Anti-human Immunodeficiency Virus Activity of the Skeleton Isomers of 3',4'-Di-(O)-(-)-camphanoyl-(+)-khellactone
Hiromi NISHIOKAa, Koji UESUGIa, Norihiro UEDAa, Yuka KONDOa, Megumi TSUJIa, Hitoshi ABEb, Takashi HARAYAMAa, Takayuki HAMASAKIc, Masanori BABAc, Yasuo TAKEUCHIa
aDivision of Pharmaceutical Sciences, Graduate School of Medicine, Dentistry and Pharmaceutical Sciences, Okayama University, bFaculty of Engineering, Toyama University, cDivision of Antiviral Chemotherapy Center for Chronic Viral Diseases Graduate School of Medical and Dental Sciences, Kagoshima University
Chemical & Pharmaceutical Bulletin 59 (8) 1075-1076, 2011.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に121円(税込) です。