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Chemical and Pharmaceutical Bulletin 65巻 10号

発行元
日本薬学会
ISSN
0009-2363
ISSN(オンライン)
1347-5223

書籍情報から探す
開始頁
Gibbs Free Energy of Hydrolytic Water Molecule in Acyl-Enzyme Intermediates of a Serine Protease : A Potential Application for Computer-Aided Discovery of Mechanism-Based Reversible Covalent Inhibitors
Yosuke Masuda, Noriyuki Yamaotsu, Shuichi Hirono
School of Pharmaceutical Sciences, Kitasato University
Chemical and Pharmaceutical Bulletin 65 (10) 889-892, 2017.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Synthesis, Docking Simulation, Biological Evaluations and 3D-QSAR Study of 1,4-Dihydropyridines as Calcium Channel Blockers
Tarek Fathy El-Moselhy(a), Peter Ayoub Sidhom(a), Eman Ahmed Esmat(a), Nageh Ahmed El-Mandy(b)
(a)Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Tanta University, (b)Department of Pharmacology, Faculty of Pharmacy, Tanta University
Chemical and Pharmaceutical Bulletin 65 (10) 893-903, 2017.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Design, Synthesis, Antifungal Activity and Molecular Docking of Thiochroman-4-one Derivatives
Yifan Zhong(a), Xiaoyan Han(a), Shengbin Li(a), Hui Qi(a), Yali Song(a),(b), Xiaoqiang Qiao(a),(b)
(a)Key Laboratory of Pharmaceutical Quality Control of Hebei Province, College of Pharmaceutical Sciences, Hebei University, (b)Key Laboratory of Medicinal Chemistry and Molecular Diagnosis of Ministry of Education, Hebei University
Chemical and Pharmaceutical Bulletin 65 (10) 904-910, 2017.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Antileishmanial Thioureas : Synthesis, Biological Activity and in Silico Evaluations of New Promising Derivatives
Gil Mendes Viana(a), Deivid Costa Soares(b), Marcos Vinicius Santana(c), Lilian Henriques do Amaral(a), Paloma Wetler Meireles(a), Raquel Pinto Nunes(a), Luiz Claudio Rodrigues Pereira da Silva(a), Lucia Cruz de Sequeira Aguiar(d), Carlos Rangel Rodrigues(e), Valeria Pereira de Sousa(a), Helena Carla Castro(c), Paula Alvarez Abreu(f), Plinio Cunha Sathler(a), Elvira Maria Saraiva(b), Lucio Mendes Cabral(a)
(a)Universidade Federal do Rio de Janeiro, LabTIF, Faculdade de Farmacia, Ilha do Fundao, (b)Universidade Federal do Rio de Janeiro, Laboratorio de Imunobiologia das Leishmanioses, Instituto de Microbiologia Paulo de Goes, (c)Universidade Federal Fluminense, LABiEMol, Departamento de Biologia Celular e Molecular, Outeiro de Sao Joao Baptista, (d)Universidade Federal do Rio de Janeiro, Instituto de Quimica, Ilha do Fundao, (e)Universidade Federal do Rio de Janeiro, ModMolQSAR, Faculdade de Farmacia, Ilha do Fundao, (f)Laboratorio de Modelagem Molecular e Pesquisa em Ciencias Farmaceuticas, LaMCiFar. Universidade Federal do Rio de Janeiro-Campus Macae
Chemical and Pharmaceutical Bulletin 65 (10) 911-919, 2017.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
C-Homomorphinan Derivatives as Lead Compounds to Obtain Safer and More Clinically Useful Analgesics
Kyoko Ishikawa(a), Fumika Karaki(a),(b), Kaoru Tayama(a), Eika Higashi(a), Shigeto Hirayama(a),(b), Kennosuke Itoh(a),(b), Hideaki Fujii(a),(b)
(a)Laboratory of Medicinal Chemistry, School of Pharmacy, Kitasato University, (b)Medicinal Research Laboratories, School of Pharmacy, Kitasato University
Chemical and Pharmaceutical Bulletin 65 (10) 920-929, 2017.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Microtropins Q-W, ent-Labdane Glucosides : Microtropiosides G-I, Ursane-Type Triterpene Diglucoside and Flavonol Glycoside from the Leaves of Microtropis japonica
Saori Terazawa(a), Yuka Uemura(a), Yuka Koyama(a), Susumu Kawakami(b), Sachiko Sugimoto(a), Katsuyoshi Matsunami(a), Hideaki Otsuka(a),(b), Takakazu Shinzato(c), Masatoshi Kawahata(d), Kentaro Yamaguchi(d)
(a)Graduate School of Biomedical and Health Sciences, Hiroshima University, (b)Faculty of Pharmacy, Yasuda Women's University, (c)Subtropical Field Science Center, Faculty of Agriculture, University of the Ryukyus, (d)Faculty of Pharmaceutical Sciences, Tokushima Bunri University, Kagawa Campus
Chemical and Pharmaceutical Bulletin 65 (10) 930-939, 2017.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Versatile Amine-Promoted Mild Methanolysis of 3,5-Dinitrobenzoates and Its Application to the Synthesis of Colorado Potato Beetle Pheromone
Yumiko Yamano, Haruna Sasaki, Akimori Wada
Department of Organic Chemistry for Life Science, Kobe Pharmaceutical University
Chemical and Pharmaceutical Bulletin 65 (10) 940-944, 2017.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Rapid Analysis of DOXIL Stability and Drug Release from DOXIL by HPLC Using a Glycidyl Methacrylate-Coated Monolithic Column
Arato Kimoto(a), Ayako Watanabe(b), Eiichi Yamamoto(c), Tatsuya Higashi(a), Masaru Kato(b)
(a)Faculty of Pharmaceutical Sciences, Tokyo University of Science, (b)Graduate School of Pharmaceutical Sciences, The University of Tokyo, (c)Formulation Research, Pharmaceutical Science and Technology, Core Function Unit, Medicine Development Center, Eisai Co.,Ltd.
Chemical and Pharmaceutical Bulletin 65 (10) 945-949, 2017.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Design, Synthesis and Antiproliferative Evaluation of Novel Disulfides Containing 1,3,4-Thiadiazole Moiety
Shuai Zhang, Xiao-jia Liu, Rui Tang, Hai-xin Wang, Hai-ying Liu, Yu-ming Liu, Bao-quan Chen
Tianjin Key Laboratory of Organic Solar Cells and Photochemical Conversion, School of Chemistry & Chemical Engineering, Tianjin University of Technology
Chemical and Pharmaceutical Bulletin 65 (10) 950-958, 2017.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Docetaxel-Loaded Lecithoid Nanoparticles with Enhanced Lung Targeting Efficiency and Reduced Systemic Toxicity : Developed by Solid Dispersion and Effervescent Techniques
Li Zhang(a), Zhong-hong Liu(a), Xun-guan Cheng(a), Zhu Xia(b), Yu Liu(c), Yu Yu(a)
(a)Research Laboratory of Medicinal Chemistry and Biomaterials, Chongqing Pharmaceutical Engineering Research Center, School of Pharmacy, Chongqing Medical University, (b)Department of Nuclear Medicine, The First Affiliated Hospital of Chongqing Medical University, (c)Department of Pharmacy, The First Affiliated Hospital of Chongqing Medical University
Chemical and Pharmaceutical Bulletin 65 (10) 959-966, 2017.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Prediction of Dissolution Data Integrated in Tablet Database Using Four-Layered Artificial Neural Networks
Kozo Takayama(a), Shota Kawai(b), Yasuko Obata(b), Hiroaki Todo(a), Kenji Sugibayashi(a)
(a)Department of Pharmaceutical Sciences, Faculty of Pharmacy and Pharmaceutical Sciences, Josai University, (b)Department of Pharmaceutical Sciences, Hoshi University
Chemical and Pharmaceutical Bulletin 65 (10) 967-972, 2017.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
5,6-Dihydropyrrolo[2,1-α]isoquinolines as Alternative of New Drugs with Cytotoxic Activity
Rosa Maria Chavez-Santos(a), Paul Eduardo Reyes-Gutierrez(b), Ruben Omar Torres-Ochoa(a), Maria Teresa Ramirez-Apan(a), Roberto Martinez(a)
(a)Instituto de Quimica, Universidad Nacional Autonoma de Mexico, Circuito Exterior, Ciudad Universitaria, (b)Institute of Organic Chemistry and Biochemistry, Czech Academy of Sciences
Chemical and Pharmaceutical Bulletin 65 (10) 973-981, 2017.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Triplex- and Duplex-Forming Abilities of Oligonucleotides Containing 2'-Deoxy-5-trifluoromethyluridine and 2'-Deoxy-5-trifluoromethylcytidine
Yuta Ito, Misaki Matsuo, Takashi Osawa, Yoshiyuki Hari
Faculty of Pharmaceutical Sciences, Tokushima Bunri University
Chemical and Pharmaceutical Bulletin 65 (10) 982-988, 2017.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Asymmetric Aldol/Vinylogous Aldol/Cyclization Reaction Using Phosphine Oxide Catalysts
Nathan Ray Alim(a), Shiki Miyazaki(a), Yasushi Shimoda(a), Masaharu Sugiura(a), Makoto Nakajima(a), Shunsuke Kotani(a),(b)
(a)Graduate School of Pharmaceutical Sciences, Kumamoto University, (b)Priority Organization for Innovation and Excellence, Kumamoto University
Chemical and Pharmaceutical Bulletin 65 (10) 989-993, 2017.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。
Affinity Labeling with 4-Azidophthalimide (AzPI) : Relation between Labeling Rate and Fluorescence Intensity
Kosuke Chiba, Yuichi Hashimoto, Takao Yamaguchi†
Institute of Molecular and Cellular Biosciences, The University of Tokyo, †Present address : Graduate School of Pharmaceutical Sciences, Osaka University
Chemical and Pharmaceutical Bulletin 65 (10) 994-996, 2017.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。