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Chemical and Pharmaceutical Bulletin 67巻 10号

発行元
日本薬学会
ISSN
0009-2363
ISSN(オンライン)
1347-5223

書籍情報から探す
開始頁
Combinatorial Synthesis and Biological Evaluation of Destruxins
Masahito Yoshida
Faculty of Pure and Applied Sciences, University of Tsukuba
Chemical and Pharmaceutical Bulletin 67 (10) 1023-1029, 2019.
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A Snapshot on the Current Status of Alzheimer's Disease, Treatment Perspectives, in-Vitro and in-Vivo Research Studies and Future Opportunities
Gizem Tezel(a), Selin Seda Timur(a), Ismail Bozkurt(b), O.Faruk Turkoglu(c), Ipek Eroglu(d), Emirhan Nemutlu(e), Levent Oner(a), Hakan Eroglu(a)
(a)Department of Pharmaceutical Technology, Faculty of Pharmacy, Hacettepe University, (b)Department of Neurosurgery, Cankiri State Hospital, (c)Department of Neurosurgery, Ankara Ataturk Research and Education Hospital, (d)Department of Basic Pharmaceutical Sciences, Faculty of Pharmacy, Hacettepe University, (e)Department of Analytical Chemistry, Faculty of Pharmacy, Hacettepe University
Chemical and Pharmaceutical Bulletin 67 (10) 1030-1041, 2019.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Tetramethylammonium Fluoride Tetrahydrate-Mediated Transition Metal-Free Coupling of Aryl Iodides with Unactivated Arenes in Air
Kanako Nozawa-Kumada, Kosuke Nakamura, Satoshi Kurosu, Yuki Iwakawa, Charline Denneval, Masanori Shigeno, Yoshinori Kondo
Graduate School of Pharmaceutical Sciences, Tohoku University
Chemical and Pharmaceutical Bulletin 67 (10) 1042-1045, 2019.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Lewis Base Assisted Lithium Bronsted Base Catalysis : A New Entry for Catalytic Asymmetric Synthesis of β2,2-Amino Acids
Fuyuki Amemiya, Hidetoshi Noda, Masakatsu Shibasaki
Institute of Microbial Chemistry, Tokyo
Chemical and Pharmaceutical Bulletin 67 (10) 1046-1049, 2019.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Development of Universal Formulation with Superior Re-dispersion Using Nanocrystal Approach with Simultaneous Identification of API Physicochemical Properties
Hiroyuki Fujii, Satoru Watano
Department of Chemical Engineering, Graduate School of Engineering, Osaka Prefecture University
Chemical and Pharmaceutical Bulletin 67 (10) 1050-1060, 2019.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Geometrical Conversion of the EGFR Extracellular Domain by Adiabatic Mapping Combining Normal Mode Analysis of the Elastic Network Model and Energy Optimization
Hiroyuki Nojima, Yasuomi Kiyota, Genki Terashi, Mayuko Takeda-Shitaka, Hajime Matsubara
School of Pharmacy, Kitasato University
Chemical and Pharmaceutical Bulletin 67 (10) 1061-1071, 2019.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Biosynthesis of Novel Shikonin Glucosides by Enzymatic Glycosylation
Bohan Li(a), Meilin Zhu(a), Hui Ma(a), Tao Ma(a), Yiqun Dai(a), Hongmei Li(a), Yu Li(b), Cheng-Zhu Wu(a)
(a)School of Pharmacy, Bengbu Medical College, (b)School of Pharmacy, Second Military Medical University
Chemical and Pharmaceutical Bulletin 67 (10) 1072-1075, 2019.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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An Improved Protocol for the Virtual Screening Discovery of Novel Histone Deacetylase Inhibitors
Qiuhang Song(a), Tingting Liu(a), Yucui Liu(b), Shuyue Wang(a), Cong Fan(c), Lihua Zheng(d), Yongli Bao(a), Luguo Sun(a), Chunlei Yu(d), Ying Sun(a), Zhenbo Song(a), Guannan Wang(d), Yanxin Huang(a), Yuxin Li(d)
(a)National Engineering Laboratory for Druggable Gene and Protein Screening, Northeast Normal University, (b)State Key Laboratory of Microbial Technology, Shandong University, (c)Sun Yat-Sen Memorial Hospital, Sun Yat-Sen University, (d)Research Center of Agriculture and Medicine gene Engineering of Ministry of Education, Northeast Normal University
Chemical and Pharmaceutical Bulletin 67 (10) 1076-1081, 2019.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Transporter-Targeted Bile Acid-Camptothecin Conjugate for Improved Oral Absorption
Linxia Xiao, Yuqin Zhou, Xiangli Zhang, Yan Ding, Qingyong Li
Collaborative Innovation Center of Yangtze River Region Green Pharmaceuticals, Zhejiang University of Technology
Chemical and Pharmaceutical Bulletin 67 (10) 1082-1087, 2019.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Synthesis and Biological Evaluation of Novel L-Homoserine Lactone Analogs as Quorum Sensing Inhibitors of Pseudomonas aeruginosa
Haoyue Liu(a),(b),(c), Qianhong Gong(d), Chunying Luo(a),(b),(c), Yongxi Liang(a),(b),(c), Xiaoyan Kong(a),(b),(c), Chunli Wu(a),(b),(c), Pengxia Feng(a),(b),(c), Qing Wang(a),(b),(c), Hui Zhang(a),(b),(c), M.A. Wireko(a),(b),(c)
(a)School of Pharmaceutical Sciences, Zhengzhou University, (b)Key Laboratory of Technology of Drug Preparation (Zhengzhou University), Ministry of Education of China, (c)Key Laboratory of Henan Province for Drug Quality and Evaluation, (d)Key Laboratory of Marine Drugs, Chinese Ministry of Education, School of Medicine and Pharmacy, Ocean University of China
Chemical and Pharmaceutical Bulletin 67 (10) 1088-1098, 2019.
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Novel Cubosome System Resistant to Lipid Removal by Serum Albumin
Makoto Uyama(a), Tetsurou Handa(b), Minoru Nakano(c)
(a)Shiseido Global Innovation Center, (b)Faculty of Pharmaceutical Sciences, Suzuka University of Medical Science, (c)Graduate School of Medicine and Pharmaceutical Sciences, University of Toyama
Chemical and Pharmaceutical Bulletin 67 (10) 1099-1103, 2019.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Comparative Metabolite Profiling of Wild and Cultivated Licorice Based on Ultra-Fast Liquid Chromatography Coupled with Triple Quadrupole-Time of Flight Tandem Mass Spectrometry
Chengcheng Wang(a), Zhichen Cai(a), Jingjing Shi(a), Shuyu Chen(a), Mengxia Tan(a), Jiali Chen(a), Lihong Chen(a), Lisi Zou(a), Cuihua Chen(a), Zixiu Liu(a), Xunhong Liu(a),(b),(c)
(a)School of Pharmacy, Nanjing University of Chinese Medicine, (b)Collaborative Innovation Center of Chinese Medicinal Resources Industrialization, (c)National and Local Collaborative Engineering Center of Chinese Medicinal Resources Industrialization and Formulae Innovative Medicine
Chemical and Pharmaceutical Bulletin 67 (10) 1104-1115, 2019.
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Design, Synthesis and Biological Evaluation of Novel Benzoylimidazole Derivatives as Raf and Histone Deacetylases Dual Inhibitors
Xin Chen(a), Guoliang Gong(a), Xinyang Chen(a), Ruihu Song(a), Mei Duan(a), Ruizhi Qiao(a), Yu Jiao(b), Jianzhao Qi(a), Yadong Chen(b), Yong Zhu(b)
(a)Shaanxi Key Laboratory of Natural Products & Chemical Biology, College of Chemistry & Pharmacy, Northwest A&F University, (b)School of Science, China Pharmaceutical University
Chemical and Pharmaceutical Bulletin 67 (10) 1116-1122, 2019.
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Effects of the 2-Substituted Adenosine-1,3-diazaphenoxazine 5'-Triphosphate Derivatives on the Single Nucleotide Primer Extension Reaction by DNA Polymerase
Yosuke Taniguchi, Ikuko Sagara, Yusuke Nagata, Yoshiya Kikukawa, Shigeki Sasaki
Graduate School of Pharmaceutical Sciences, Kyushu University
Chemical and Pharmaceutical Bulletin 67 (10) 1123-1130, 2019.
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Development of a Membrane Curvature-Sensing Peptide Based on a Structure-Activity Correlation Study
Kenichi Kawano, Masaya Ogushi, Toshihiro Masuda, Shiroh Futaki
Institute for Chemical Research, Kyoto University
Chemical and Pharmaceutical Bulletin 67 (10) 1131-1138, 2019.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Non-naturally Occurring Helical Molecules Can Interfere with p53-MDM2 and p53-MDMX Protein-Protein Interactions
Aoze Su(a), Siyuan Wang(a), Akane Sada(b), Yuko Otani(a), Luhan Zhai(a), Xin Liu(a), Misa Sayama(a), Rieko Ohki(b), Tomohiko Ohwada(a)
(a)Graduate School of Pharmaceutical Sciences, University of Tokyo, (b)Laboratory of Fundamental Oncology, National Cancer Center Research Institute
Chemical and Pharmaceutical Bulletin 67 (10) 1139-1143, 2019.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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The Usefulness of Definitive Screening Design for a Quality by Design Approach as Demonstrated by a Pharmaceutical Study of Orally Disintegrating Tablet
Keisuke Takagaki(a), Terushi Ito(b), Hiroaki Arai(a), Yasuko Obata(a), Kozo Takayama(c), Yoshinori Onuki(b)
(a)Department of Pharmaceutics, Hoshi University, (b)Laboratory of Pharmaceutical Technology, Graduate School of Medical and Pharmaceutical Science, University of Toyama, (c)Faculty of Pharmacy and Pharmaceutical Sciences, Josai University
Chemical and Pharmaceutical Bulletin 67 (10) 1144-1151, 2019.
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Controlled-Release Fine Particles Prepared by Melt Adsorption for Orally Disintegrating Tablets
Kai Shiino(a),(b), Takao Oshima(a), Ryoichi Sonoda(a), Shin-ichiro Kimura(b), Shigeru Itai(b), Yasunori Iwao(b)
(a)Formulation Department, CMC center, Kaken Pharmaceutical Co., Ltd., (b)Department of Pharmaceutical Engineering, School of Pharmaceutical Sciences, University of Shizuoka
Chemical and Pharmaceutical Bulletin 67 (10) 1152-1159, 2019.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
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Chemometric Evaluation of Repeatability Using the Autocorrelation Method in High-Performance Liquid Chromatography with Ultraviolet Detection
Akira Kotani(a), Mitsuo Saito(a),(b), Takehiko Yajima(b), Hideki Hakamata(a), Yuzuru Hayashi(b),(c)
(a)School of Pharmacy, Tokyo University of Pharmacy and Life Sciences, (b)Institute for Health Vigilance, (c)Institute of FUMI Theory
Chemical and Pharmaceutical Bulletin 67 (10) 1160-1163, 2019.
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Reactions of Rebamipide with Hypobromous Acid
Toshinori Suzuki, Akane Okuyama
School of Pharmacy, Shujitsu University
Chemical and Pharmaceutical Bulletin 67 (10) 1164-1167, 2019.
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Adsorption Capability of Fe-HT3.0 for Nitrite and Nitrate Ions in a Binary Solution System
Fumihiko Ogata(a), Noriaki Nagai(a), Takehiro Nakamura(a), Naohito Kawasaki(a),(b)
(a)Faculty of Pharmacy, Kindai University, (b)Antiaging Center, Kindai University
Chemical and Pharmaceutical Bulletin 67 (10) 1168-1170, 2019.
  • アブストラクト: 従量制は110円(税込)、基本料金制は基本料金に含まれます。
  • 全文ダウンロード: 従量制、基本料金制の方共に770円(税込) です。