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BCSクラスIII薬物(ラニチジン)のバイオアベイラビリティに対するポリエチレングリコール400(PEG400)の影響 Polyethylene glycol 400 enhances the bioavailability of a BCS class III drug(ranitidine) in male subjects but not females Ashiru DA, et al:Pharm Res, 25(10):2327-2333, 2008
取り込みおよび排出トランスポーターが関与するセリプロロールの消化管吸収 Involvement of influx and efflux transport systems in gastrointestinal absorption of celiprolol Kato Y, et al:J Pharm Sci, 9 Dec 2008 DOI(10.1002/jps.21618)
Glyburideの体内動態と血糖低下作用に対するリファンピシンの誘導と阻害の影響 Elucidating rifampin's inducing and inhibiting effects on glyburide pharmacokinetics and blood glucose in healthy volunteers:unmasking the differential effects of enzyme induction and transporter inhibition for a drug and its primary metabolite Zheng HX, et al:Clin Pharmacol Ther, 85:78-85, 2009
チオールアダクト体生成による50薬剤のin vitroスクリーニング ―特異体質性毒性と共有結合生成量との比較 In vitro screening of 50 highly prescribed drugs for thiol adduct formation: comparison of potential for drug-Induced toxicity and extent of adduct formation Gan J, et al:Chem Res Toxicol, Article ASAP, published on 02 March 2009